Studies on New β-Adrenergic Blocking Agents. II. Syntheses and Pharmacology of 2-Anilinotropone Derivatives
スポンサーリンク
概要
- 論文の詳細を見る
2-[p-(Aminoalkoxy) anilino] tropone derivatives were prepared from 2-(p-hydroxyanilino) tropone derivatives by established synthetic procedures and were tested for β-adrenergic blocking, coronary vasodilating, and anti-hypertensive activities. Some members of the series exhibited significant activities in one or more of the pharmacological tests, and introduction of a halogen atom into the 5-position of the tropone nucleus caused generally an increase in the pharmacological activities.
- 社団法人日本薬学会の論文
- 1974-03-25
著者
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高木 弘
Central Research Laboratories Sankyo Co. Ltd.
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佐藤 裕信
Central Research Laboratories Sankyo Co. Ltd.
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佐藤 裕信
三共株式会社中央研究所
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小池 博之
三共株式会社中央研究所
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田中 輝夫
Central Research Laboratories, Sankyo Co., Ltd.
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熊倉 清次
Central Research Laboratories, Sankyo Co., Ltd.
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小池 博之
Central Research Laboratories, Sankyo Co., Ltd.
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大島 武史
Central Research Laboratories, Sankyo Co., Ltd.
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遠藤 和夫
Central Research Laboratories, Sankyo Co., Ltd.
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熊倉 清次
三共株式会社中央研究所
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田中 輝夫
Central Research Laboratories Sankyo Co. Ltd.
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遠藤 和夫
三共株式会社中央研究所
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大島 武史
And Biological Research Laboratories:sankyo Co. Ltd.
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