SYNTHESIS OF A NEW POTENT ANTI-ULCER AND GASTRIC SECRETORY INHIBITING AGENT, (-)-cis-2,3-DIHIDRO-3-(4-METHYLPIPERAZINYLMETHYL)-2-PHENYL-1,5-BENZOTHIAZEPIN-4 (5H)-ONE HYDROCHLORIDE (BTM-1086), AND RELATED COMPOUNDS
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概要
- 論文の詳細を見る
(-)-cis-2,3-Dihydro-3-(4-methylpiperazinylmethyl)-2-phenyl-1,5-benzothiazepin-4 (5H)-one hydrochloride (BTM-1086) and its analogues, which possessed potent anti-ulcer and gastric secretory inhibiting activities, were synthesized and the structures of these compounds were established on the basis of spectral and chemical evidences.
- 公益社団法人日本薬学会の論文
- 1983-05-25
著者
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堀 幹夫
Gifu Pharmaceutical University
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大野 左千雄
Research Laboratories, Maruko Seiyaku Co., Ltd.,
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水越 清史
Research Laboratories, Maruko Seiyaku Co., Ltd.,
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水越 清史
Research Laboratories Maruko Seiyaku Co. Ltd.
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泉 喜八郎
Research Laboratories, Maruko Pharmaceutical Co., Ltd.,
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加藤 和雄
Research Laboratories, Maruko Pharmaceutical Co., Ltd.,
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加藤 和雄
Research Laboratories Maruko Pharmaceutical Co. Ltd.
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大野 左千雄
Research Laboratories Maruko Seiyaku Co. Ltd.
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大野 佐千雄
Research Laboratories Maruko Pharmaceutical Co. Ltd.
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泉 喜八郎
Research Laboratories Maruko Pharmaceutical Co. Ltd.
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