A MODIFIED MANNICH REACTION USING 1,3-DIOXOLANE
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概要
- 論文の詳細を見る
Mannich reaction of ketones using 1,3-dioxolane instead of formaldehyde, paraformaldehyde, or 1,3,5-trioxane afforded the corresponding Mannich bases in high yields. Under the same conditions the aminomethylation of aromatics did not proceed but the intramolecular aminomethylation, like a Pictet-Spengler type reaction, proceeded smoothly.
- 公益社団法人日本薬学会の論文
- 1994-08-15
著者
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隅田 師玄
Research Laboratories, Maruko Seiyaku Co., Ltd.,
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孝森 昌幸
Research Laboratories, Maruko Seiyaku Co., Ltd.,
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孝森 昌幸
Research Laboratories Maruko Seiyaku Co. Ltd.
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大野 佐千雄
Research Laboratories Maruko Pharmaceutical Co. Ltd.
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隅田 師玄
Research Laboratories Maruko Pharmaceutical Co. Ltd.
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- A MODIFIED MANNICH REACTION USING 1,3-DIOXOLANE