Glutathione-dependent Degradation of Organophosphate Insecticides by Organophosphate-susceptible and Resistant Housefly Abdomen Homogenates
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概要
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The glutathione (GSH)-dependent degradation of salithion, which is one of the effective insecticides against Organophosphate (OP)-resistant housefly (Musca domestica L.), and that of the ineffective insecticides, fenitrothion and malathion, was studied. The most degradable insecticide was malathion (22% and 97% with susceptible SRS and OP-resistant 3-Y homogenates, respectively), then fenitrothion (9% and 26%), and the least was salithion (3% and 9%). Ethacrynic acid inhibited the in vitro degradation of all three OP-insecticides by both SRS and 3-Y homogenates, and lowered the degradation level to the same as that existing under conditions without the addition of GSH. 2-Methylthio-l, 3, 2-benzodioxaphosphorin 2-oxide, a thiolo-isomer of salithion, and O, O-diisopropyl S-ring-hydroxy-benzyl phosphorothiolates (hydroxy IBPs) inhibited the degradation of fenitrothion. The former also inhibited the carboxylesterase-dependent degradation of malathion.
- 社団法人 日本農芸化学会の論文
著者
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Shiotsuki Takahiro
Department Of Insect Physiology And Behavior National Institute Of Sericultural And Entomological Sc
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Takeya Ryuko
Department Of Agricultural Chemistry Faculty Of Agriculture Kyushu University
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Eto Morifusa
Department Of Agricultural Chemistry Faculty Of Agriculture Kyushu University
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