Synthesis of 2,2-Diphenylpropionate Derivatives and Their Effects on Larval Growth of the Silkworm

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概要

• 論文の詳細を見る

• A variety of 2,2-diphenylpropionate derivatives with an amino substituent were synthesized and their effects on larval growth of the silkworm, Bombyx mori, were examined by dietary administration. Of the compounds tested, 3- (4-ethylpiperazin-1-yl) propyl 2,2-diphenylpropionate (3) caused significant prolongation of the larval period. Studies on the structure-activity relationship indicate that a piperazine ring and the bond distances between the nitrogen atom and the ester group were important for this activity. Treatment of compound 3 delayed the increase of ecdysteroid titers in the hemolymph by 3 days compared with that of the control, which correlates with the delay in molting.

• 社団法人日本農芸化学会の論文
• 2000-03-23

著者

• SHIOTSUKI Takahiro

  Department of Insect Physiology and Behavior, National Institute of Sericultural and Entomological S

• Kuwano Eiichi

  Laboratory of Pesticide Chemistry,Division of Plant Protection,Department of Applied Genetics and Pe

• Kim In-hae

  Laboratory Of Pesticide Chemistry Department Of Applied Genetics And Pest Management Faculty Of Agri

• Kuwano Eiichi

  Laboratory Of Pesticide Chemistry Division Of Bioresource And Bioenvironmental Sciences Graduate Sch

• Kuwano Eiichi

  Laboratory Of Pesticide Chemistry Department Of Agricultural Chemistry Kyushu University

• Shiotsuki Takahiro

  Department Of Insect Physiology And Behavior National Institute Of Sericultural And Entomological Sc

• TOYOMURA Nozomu

  Laboratory of Pesticide Chemistry, Division of Bioresource and Bioenvironmental Sciences, Graduate S

• KIM InHae

  Laboratory of Pesticide Chemistry, Division of Bioresource and Bioenvironmental Sciences, Graduate S

• YOSHIDA Tetsuya

  Laboratory of Pesticide Chemistry, Division of Bioresource and Bioenvironmental Sciences, Graduate S

• Kim Inhae

  Laboratory Of Pesticide Chemistry Division Of Bioresource And Bioenvironmental Sciences Graduate Sch

• Toyomura Nozomu

  Laboratory Of Pesticide Chemistry Division Of Bioresource And Bioenvironmental Sciences Graduate Sch

• Toyomura Nozomu

  Laboratory Of Pesticide Chemistry Department Of Agricultural Chemistry Kyushu University

• Yoshida Tetsuya

  Laboratory Of Pesticide Chemistry Division Of Bioresource And Bioenvironmental Sciences Graduate Sch

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