Biological Activity of Optically Active Salithion and Salioxon
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概要
- 論文の詳細を見る
Salioxon enantiomers were obtained from salithion enantiomers by MCPBA oxidation. The larvicidal and adulticidal activities of salithion enantiomers, and the anti-cholinesterase activity of salioxon enantiomers were determined on house flies. On larvae, the potency of (S)(-)-salithion (LC50=1.1 ppm) was about two-fold higher than the (R)(+)-enantiomer (LC50 = 2.1 ppm). A similar ratio was obtained when these compounds were applied topically to female adults. The relative potency of these enantiomers correlated well with the anti-cholinesterase activity of their respective oxidative enantiomers, (R)(+)-and (S)(-)-salioxon, which are assumed to have been formed after their application to the insects.
- 社団法人 日本農芸化学会の論文
著者
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HIRASHIMA Akinori
Department of Agricultural Chemistry, Kyushu University
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Wu Shao-yong
Department Of Agricultural Chemistry Kyusyu University
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Ueno Ryohei
Department Of Agricultural Chemistry Kyushu University
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Hirashima Akinori
Department Of Agricultural Chemistry Kyushu University
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Eto Morifusa
Department Of Agricultural Chemistry Faculty Of Agriculture Kyushu University
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WU Shao-Yong
Department of Agricultural Chemistry, Kyushu University
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ISHAAYA Isaac
Department of Agricultural Chemistry, Kyushu University
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ICHIYAMA Yoshifumi
Department of Agricultural Chemistry, Kyushu University
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