Synthesis and Insect Growth Regulatory Activity of 1,5-Disubstituted Imidazoles with Non-terpene Chains(Pesticide Chemistry)

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概要

• 論文の詳細を見る

• 1-Isobutyl-5-(4-phenoxyphenyl)imidazole (KK-98), an inhibitor of juvenile hormone (JH) biosynthesis in the cockroach, and related imidazole compounds were evaluated against silkworm, Bombyx mori, for their activity to induce precocious metamorphosis. KK-98 induced precocious metamorphosis in the 4th instar larvae at high doses. Replacement of the 4-phenoxy group by a 3-phenoxy or 3-benzyloxy group on the benzene ring increased the activity. Among this series of compounds, 5-(3-benzyloxyphenyl)-1-isopropylimidazole (8) showed the highest activity. The induction of precocious metamorphosis by compound 8 was rescued by the simultaneous application of methoprene, a JH minic. When newly molted 3rd instar larvae were treated with a high dose of compound 8, a few larvae formed larval-pupal intermediates in the 3rd instar stage, which has not been formed by treating of any other imidazoles so far.

• 社団法人日本農芸化学会の論文
• 1991-12-23

著者

• KUWANO Eiichi

  Department of Agricultural Chemistry, Kyushu University

• ETO Morifusa

  Department of Agricultural Chemistry, Kyushu University

• Eto Morifusa

  Department Of Agricultural Chemistry Kyushu University

• Kuwano Eiichi

  Department Of Agricultural Chemistry Faculty Of Agriculture Kyushu University

• Kuwano E

  Kyushu Univ. Fukuoka Jpn

• Hisano Tomomi

  Department of Agricultural Chemistry, Kyushu University

• Eto Morifusa

  Department Of Agricultural Chemistry Faculty Of Agriculture Kyushu University

• Hisano Tomomi

  Department Of Agricultural Chemistry Kyushu University

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