Comparative Characterization of Lung Muscarinic Receptor Binding After Intratracheal Administration of Tiotropium, Ipratropium, and Glycopyrrolate

スポンサーリンク

概要

• 論文の詳細を見る
• 2011-03-20

著者

• Yamada Shizuo

  Dep. Of Pharmacokinetics And Pharmacodynamics And Global Center Of Excellence (coe) Program School O

• Yamada Shizuo

  Department Of Biophamacy School Of Pharmaceutical Sciences University Of Shizuoka

• OGODA Masaki

  Department of Pharmacokinetics and Pharmacodynamics and Global Center of Excellence (COE) Program, S

• NIIYA Ryo

  Department of Pharmacokinetics and Pharmacodynamics and Global Center of Excellence (COE) Program, S

• KOSHIKA Tadatsura

  Pharmacology Research Laboratories, Drug Discovery Research, Astellas Pharma Inc.

• Niiya Ryo

  Department Of Pharmacokinetics And Pharmacodynamics And Global Center Of Excellence (coe) Program Sc

• Ogoda Masaki

  Department Of Pharmacokinetics And Pharmacodynamics And Global Center Of Excellence (coe) Program Sc

• Koshika Tadatsura

  Pharmacology Research Laboratories Drug Discovery Research Astellas Pharma Inc.

関連論文

• The Forefront for Novel Therapeutic Agents Based on the Pathophysiology of Lower Urinary Tract Dysfunction: Bladder Selectivity Based on In Vivo Drug–Receptor Binding Characteristics of Antimuscarinic Agents for Treatment of Overactive Bladder
• Pharmacologically Relevant Receptor Binding Characteristics and 5α-Reductase Inhibitory Activity of Free Fatty Acids Contained in Saw Palmetto Extract(Pharmacology)
• Effects of Dietary Ingredients on Function and Expression of P-Glycoprotein in Human Intestinal Epithelial Cells
• Structure-Activity Relationships of Receptor Binding of 1,4-Dihydropyridine Derivatives(Pharmacology)
• PJ-566 Influence of CYP2C9 Genotype on Pharmacokinetics and Pharmacodynamics of Benzbromarone(Cardiovascular pharmacology, basic/clinical-6, The 71st Annual Scientific Meeting of the Japanese Circulation Society)
• Comparative Evaluation of Exocrine Muscarinic Receptor Binding Characteristics and Inhibition of Salivation of Solifenacin in Mice(Pharmacology)
• Isolation and Pharmacological Characterization of Fatty Acids from Saw Palmetto Extract
• Highly Sensitive Measurement of P-Glycoprotein-Mediated Transport Activity in Caco-2 Cells
• Relationship between Development of Nephrotoxicity and Blood Concentration of Cyclosporine A in Bone-Marrow Transplanted Recipients Who Received the Continuous Intravenous Infusion(Pharmacology)
• Enhancement by Grapefruit Juice of Morphine Antinociception(Pharmacology)
• Antinociceptive Effects of St. John's Wort, Harpagophytum Procumbens Extract and Grape Seed Proanthocyanidins Extract in Mice(Pharmacology)
• The 5-HT_2 Receptor Antagonist Reduces Immobility of Mice Treated with the Atypical Antidepressant Mianserin in the Forced Swimming Test
• Development of a New Vasoactive Intestinal Peptide Analogue and Its Topical Administration System, Dry Powder Inhalation
• The Structural Biology of VIP (2) : Biological Activity of VIP is Dependent on its Secondary Structure
• Prediction of α_1-Adrenoceptor Occupancy in the Human Prostate from Plasma Concentrations of Silodosin, Tamsulosin and Terazosin to Treat Urinary Obstruction in Benign Prostatic Hyperplasia(Pharmacology)
• EFFECT OF PIPERIDINE AND RELATED ALICYCLIC AMINES ON NICOTINIC AND MUSCARINIC AGONIST BINDING SITES IN THE MAMMALIAN BRAIN
• P-253 DEVELOPMENT OF POTENT HISTAMINE H_3 AND/OR H_4 RECEPTOR ANTAGONISTS BY THE STEREOCHEMICAL DIVERSITY-ORIENTED CONFORMATIONAL RESTRICTION STRATEGY
• Synthesis of Conformationally Restricted Analogs of Baclofen, a Potent GABA_B Receptor Agonist, by the Introduction of a Cyclopropane Ring
• Low Dosage of Streptozotocin and Fat-diet Reduced Rat Liver Insulin Receptor Activities
• Evaluation on Rat Model of Metabolic Syndrome Induced by Fat-diet and Streptozotocin
• RATIONALE FOR THE USE OF α-BLOCKERS IN THE TREATMENT OF BENIGN PROSTATIC HYPERPLASIA (BPH)
• In Vivo Measurement of 1, 4-Dihydropyridine Receptors in Mesenteric Arteries of Spontaneously Hypertensive Rats and Effect of Nifedipine and Cilnidipine
• Muscarinic Receptor Binding Characteristics in Rat Tissues after Oral Administration of Oxybutynin and Propiverine
• Improvement in the Histopathology of Hearts from Cardiomyopathic BIO TO-2 Hamsters Following Long-Term Administration of Amlodipine and Cilnidipine
• Ex Vivo and in Vivo α_1-Adrenoceptor Binding Characteristics of a Novel α_-Adrenoceptor Antagonist, JTH-601,in Rat Tissues
• Comparative Study on Pharmacokinetics and in Vivoα_1-Adrenoceptor Binding of [^3H]Tamsulosin and [^3H]Prazosin in Rats
• Onset of Clinical Effects and Plasma Concentration of Fluvoxamine in Japanese Patients
• Effects of Cigarette Smoking and Cytochrome P450 2D6 Genotype on Fluvoxamine Concentration in Plasma of Japanese Patients
• Time-Dependent Induction of Hepatic Cytochrome P450 Enzyme Activity and mRNA Expression by Bilobalide in Rats
• Nasal Absorption of Digoxin in Rats
• Comparative Characterization of Lung Muscarinic Receptor Binding After Intratracheal Administration of Tiotropium, Ipratropium, and Glycopyrrolate
• HYPO-ACTIVITY OF LIVER INSULIN RECEPTOR IN GOTO-KAKISAKI RATS IMPROVED BY NATURAL VANADIUM CONTANING WATER(Endocrinology,Abstracts of papers presented at the 74^ Annual Meeting of the Zoological Society of Japan)
• Characterization of Specific[^3H]Nociceptin Binding in Rat Brain and Spinal Cord
• Effects of Repeated Morphine Treatment on the Antinociceptive Effects, Intestinal Absorption, and Efflux from Intestinal Epithelial Cells of Morphine
• THE INFLUENCE OF EXTRACELLULAR Ca2+ CONCENTRATION ON THE INHIBITORY EFFECT OF ADENOSINE IN GUINEA-PIG ILEAL LONGITUDINAL MUSCLES
• Pharmacokinetic and Pharmacodynamic Analysis of Acetylcholinesterase Inhibition by Distigmine Bromide in Rats
• Demonstration of Muscarinic and Nicotinic Receptor Binding Activities of Distigmine to Treat Detrusor Underactivity
• Benzbromarone Pharmacokinetics and Pharmacodynamics in Different Cytochrome P450 2C9 Genotypes
• COMPARATIVE STUDIES ON ANTI-NICOTINIC ACTION OF HEXAMETHONIUM, MECAMYLAMINE AND ADENOSINE IN THE GUINEA PIG ISOLATED ILEUM
• EFFECTS OF SURUGATOXIN ON ADRENERGICALLY INNERVATED TISSUES
• The Forefront for Novel Therapeutic Agents Based on the Pathophysiology of Lower Urinary Tract Dysfunction : Bladder Selectivity Based on In Vivo Drug-Receptor Binding Characteristics of Antimuscarinic Agents for Treatment of Overactive Bladder
• Comparative Characterization of Lung Muscarinic Receptor Binding After Intratracheal Administration of Tiotropium, Ipratropium, and Glycopyrrolate
• EFFECT OF PICROTOXIN ON ADRENAL CATECHOLAMINE SECRETION
• EFFECTS OF NICOTINIC RECEPTOR AGONISTS AND ANTAGONISTS ON UPTAKE AND EFFLUX OF 45Ca IN PERFUSED BOVINE ADRENAL GLANDS
• Effects of Functional Food Constituents on P-glycoprotein Activity in Caco-2 Cells Determined by a New Method Using Confocal Laser Scanning Microscopy
• Inhibitory Effects of Citrus Polymethoxyflavones, Nobiletin and its Analogues, on Acetylcholinesterase Activity
• A simple method to evaluate reactivity of acylglucuronides optimized for early stage drug discovery
• Beneficial Effects of Gosha-jinki-gan and Green Tea Extract in Rats With Chemical Cystitis
• Plasma Concentration and Occupation of Calcium (Ca2+) Antagonist Receptors of Amlodipine, a Long-acting Ca2+ Antagonist in SHR
• Muscarinic Receptor Binding of the Novel Radioligand, [3H]Imidafenacin in the Human Bladder and Parotid Gland
• Bladder Endothelin-1 Receptor Binding of Bosentan and Ambrisentan
• Alterations in Renal α and β-Adrenoceptors in Stroke-Prone Spontaneously Hypertensive Rats (SHRSP)
• Inhibition by chlorpromazine, metals and I-ascorbic acid of calcium-ATPase and magnesium-ATPase in bovine adrenal medullary microsomes.
• Reduced .ALPHA.2-adrenoceptor binding in lower brainstem of stroke-prone spontaneously hypertensive rats.
• Reciprocal alteration in cardiac and hypothalamic adrenergic receptors in spontaneously hypertensive rats
• Central Acetylcholine Receptors in Spontaneously Hypertensive Rats
• Effect of 2,4,6-trinitrophenol on catecholamine secretion from perfused bovine adrenal glands.
• Determination of the Effects of Green Tea Extract and Fruit Extracts on P-glycoprotein Activity in Caco-2 Cells by Using a New Method Involving Confocal Laser Scanning Microscopy

もっと見る 閉じる

スポンサーリンク