A New Synthesis of the Aporphine Alkaloids (±)-Glaucine and(±)-Nantenine. Application of [3C + 3C] Annelation to the D-Ring Formation
スポンサーリンク
概要
- 論文の詳細を見る
A [3C + 3C] annelation using 1,1-bis(ethulthio)-2-propanone was applied to a new synthesis of the aporphine alkaloids. Condensation of the ketone with the Mannich base gave two isomeric cyclohexenones, which were converted into the aporphine framework by aromatization. (±)-Glaucine and (±)-nantenine were prepared by employing this new aromatic synthesis.
- 社団法人日本薬学会の論文
- 1993-03-15
著者
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尾崎 裕
城西大学薬学部
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尾崎 裕
Faculty Of Pharmaceutical Sciences Osaka University
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金 相元
城西大学薬学部
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久保 綾子
Faculty of Pharmaceutical Sciences, Josai University
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金 相元
Faculty of Pharmaceutical Sciences, Josai University
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金 相元
Faculty Of Pharmaceutical Sciences Josai University
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Ozaki Y
Division Of Pharmacognosy And Phytochemistry National Institute Of Health Sciences
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Ozaki Y
National Inst. Health Sci. Tokyo Jpn
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Kubo A
Meiji Pharmaceutical University
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久保 綾子
Faculty Of Pharmaceutical Sciences Josai University
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