A Convenient Synthesis of Toxoflavins, Toxoflavin 4-Oxides and 1-Demethyltoxoflavins
スポンサーリンク
概要
- 論文の詳細を見る
A convenient synthesis of toxoflavins and toxoflavin 4-oxides, which consists of the nitrosative cyclization of the aldehyde hydrazones of 3-methyl-6-(1-methylhydrazino) uracil, is described. Both toxoflavins and toxoflavin 4-oxides gave the corresponding 1-demethyltoxoflavins (8-demethylfervenulins) by treatment with nucleophiles such as dimethylformamide, dimethylacetamide and acetic acid. The preparation of some 4,8-dihydrotoxoflavin derivatives is described.
- 公益社団法人日本薬学会の論文
- 1975-09-25
著者
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米田 文郎
Faculty Of Pharmaceutical Sciences Kyoto University
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永松 朝文
Faculty Of Pharmaceutical Sciences Okayama University
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