An Improved Synthesis of optically Active Steroids
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概要
- 論文の詳細を見る
17α-Hydroxy-3-methoxy-8,14-secoestra-1,3,5(10), 9-tetraen-14-one(IIa) which is an intermediate for the total synthesis of estrogens has been optically resolved. The isomer which has unnatural configuration at C-13 has been converted to estrapentaene 3-methyl ether (IVa) via the 9,14-epoxy intermediates (XI, XII, XIII, XV).
- 社団法人日本薬学会の論文
- 1973-01-25
著者
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平賀 謙太郎
武田薬品工業株式会社中央研究所
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平賀 謙太郎
Chemical Research Laboratories Research & Development Division Takeda Chemical Industries Ltd.
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三木 卓一
武田薬品工業株式会社中央研究所
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三木 卓一
Chemical Research Laboratories, Central Research Division, Takeda Chemical Industries, Ltd.
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朝子 典彦
Chemical Research Laboratories, Central Research Division, Takeda Chemical Industries, Ltd.
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