16-エチル置換ステロイドの全合成
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概要
- 論文の詳細を見る
rac-16β-Ethyl-19-nortestosterone (XI) was synthesized in 7 steps starting from 2-methyl-4-ethylcyclopentane-1,3-dione (I) and 6-methoxy-1-vinyl-1-tetralol (II). The intermediates are the mixture of 16α and 16β isomers. XI showed a strong antiandrogenic activity.
- 社団法人日本薬学会の論文
- 1973-05-25
著者
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