Total Synthesis of Pyrrolnitrin. VI. Synthesis of Nitro-chloro-2-aminoacetophenones and 1-Aryl-1,3-butanediones
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概要
- 論文の詳細を見る
Synthetic methods of nitro-chloro-2-aminoacetophenones (XV) and 1-(nitro-chlorophenyl)-1,3-butanediones (XXIII : R=H), starting materials for the synthesis of pyrrolnitrin (I) and its related compounds, were investigated. Neber rearrangement was shown to be suitable for the preparation of XV. Cleavage of ethyl 2-(nitro-chlorobenzoyl)-acetoacetate (XXI) and 2,4-pentanedione (XXII) led to XXIII (R=H).
- 社団法人日本薬学会の論文
- 1969-03-25
著者
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海尾 澄則
Research Laboratories, Fujisawa Pharmaceutical Co., Ltd.
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刈米 和夫
Research Laboratories, Fujisawa Pharmaceutical Co., Ltd.
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田中 邦彦
Research Laboratories, Fujisawa Pharmaceutical Co., Ltd.
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野口 英世
Research Laboratories, Fujisawa Pharmaceutical Co., Ltd.
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野口 英世
Research Laboratories Fujisawa Pharmaceutical Co. Ltd.
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野口 英世
藤沢薬品工業株式会社中央研究所
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田中 邦彦
Research Laboratories Fujisawa Pharmaceutical Co. Ltd.
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刈米 和夫
Research Laboratories Fujisawa Pharmaceutical Co. Ltd.
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海尾 澄則
Fujisawa Pharmaceutical Co. Ltd.
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荻野 隆
Research Laboratories Fujisawa Pharmaceutical Co. Ltd.
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