Concise Synthesis of Heterocycle-Fused Naphthoquinones by Employing Sonogashira Coupling and Tandem Addition-Elimination/Intramolecular Cyclization
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概要
- 論文の詳細を見る
A concise method for the synthesis of heterocycle-fused naphthoquinones such as naphtho[2,3-b]-furan-4,9-dione, 1H-benz[f]indole-4,9-dione, and naphtho[2,3-b]thiophene-4,9-dione was developed. This method employed Sonogashira coupling and tandem addition-elimination/intramolecular cyclization, and it enabled the preparation of versatile heterocycle-fused naphthoquinones from one substrate.
- 公益社団法人 日本薬学会の論文
著者
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Tokuda Harukuni
Department Of Biochemistry And Molecular Biology Kyoto Prefectural University Of Medicine
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Ueda Kazunori
School of Agriculture, Kinki University
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Sakaguchi Koichi
School of Agriculture, Kinki University
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Iida Akira
School of Agriculture, Kinki University
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Tokuda Harukuni
Department of Complementary and Alternative Medicine R&D, Graduate School of Medical Science, Kanazawa University
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Yamashita Mitsuaki
School of Agriculture, Kinki University
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