Rearrangement of Sulfonamide Derivatives. V. Syntheses of Methyl α-Phenyl-2- and 4-piperidineacetate.
スポンサーリンク
概要
- 論文の詳細を見る
Heating of N-phenylacetyl-2- and 4-pyridinesulfonamide 1-oxides in 10% sodium hydroxide at 90〜95°caused rearrangement reaction to form α-phenyl-2- and 4-pyridineacetic acid 1-oxides respectively. Their respective esterification and catalytic reduction with platinum-catalyst gave the hydrochloride of methyl 2- and 4-piperidineacetate and ethyl 2-piperidineacetate.
- 公益社団法人日本薬学会の論文
- 1964-05-25
著者
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内藤 武男
Central Research Laboratory, Daiichi Seiyaku Co., Ltd.
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堂森 廉三
Central Research Laboratory, Daiichi Seiyaku Co., Ltd.
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固武 竜雄
Central Research Laboratory Daiichi Seiyaku Co. Ltd.
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堂森 廉三
Research Institute Daiichi Seiyaku Co. Ltd.
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堂森 廉三
Central Research Laboratory Daiichi Seiyaku Co. Ltd.
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