Studies on Nucleosides and Nucleotides. XII. Syntheses of 3'-Amino-3'-deoxypentofuranosylcytosines

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概要

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• 1-(3'-Amino-3'-deoxy-β-D-arabinofuranosyl) cytosine derivatives (IX), (X), and (XI) were prepared from 1-(3'-azido-3'-deoxy-β-D-arabinofuranosyl) uracil (III) via 4-thiouracil derivative (VII). Attempts to prepare 2', 3'-epoxide (XVII) of down-configuration from di-O-mesyl derivative (XVI) with sodium hydroxide was failed and instead 2,2'-anhydronucleoside (XVIII) was obtained.

• 公益社団法人日本薬学会の論文
• 1969-06-25

著者

• 小林 利彦

  Central Research Laboratory Daiichi Seiyaku Co. Ltd.

• 内藤 武男

  Central Research Laboratory, Daiichi Seiyaku Co., Ltd.

• 平田 三四司

  Central Research Laboratory, Daiichi Seiyaku Co., Ltd.

• 内藤 武男

  Research Laboratories, Daiichi Seiyaku Co., Ltd.

• 内藤 武男

  Research Laboratories Daiichi Seiyaku Co. Ltd.

• 平田 三四司

  Research Institute, Daiichi Seiyaku Co., Ltd.

• 平田 三四司

  Research Institute Daiichi Seiyaku Co. Ltd.

• 平田 三四司

  Central Research Laboratory Daiichi Seiyaku Co. Ltd.

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