Synthetic Antibacterials. II. Synthesis of Pyrido [2,3-d] pyrimidine Derivatives. (1)

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概要

• 論文の詳細を見る

• The condensation of 4-substituted 6-amino-2-methylpyrimidines with diethyl ethoxymethylenemalonate, followed by thermal cyclization in Dowtherm A, yielded the corresponding 4-substituted 2-methyl-5-hydroxypyrido [2,3-d] pyrimidine-6-carboxylates. These latter compounds served as starting materaials for several transformation reactions.

• 公益社団法人日本薬学会の論文
• 1970-07-25

著者

• 千賀 慶太郎

  慶応大 病院

• 千賀 慶太郎

  慶応義塾大学病院薬剤部

• 米田 文郎

  Pharmaceutical Sciences, Kumamoto University

• 深沢 信乃夫

  Pharmaceutical Institute, School of Medicine, Keio University

• Machida Yoshiharu

  Pharmaceutical Institute School Of Medicine Keio University

• 西垣 貞男

  Pharmaceutical Institute School Of Medicine Keio University

• 西垣 貞雄

  Pharmaceutical Institute School Of Medicine Keio University

• AIDA KYOKO

  Hoshi College of Pharmacy

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