The Synthesis and Reactions of Some Isoxazolo [3,4-d] pyrimidines
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概要
- 論文の詳細を見る
The reaction of 6-hydroxyamino-1,3-dimethyluracil (1) with Vilsmeier reagent (phosphorus oxychloride and dimethylformamide) or arylaldehydes afforded 5,7-dimethyl-isoxazolo [3,4-d] pyrimidine-4,6 (5H, 7H)-dione (2) and its 3-aryl derivatives (10-17), respectively. The 3-arylisoxazolo [3,4-d] pyrimidines (9,10) underwent photorearrangement to yield the corresponding 2-aryloxazolo [4,5-d] pyrimidines (19-20). Some reactions on 2 are also reported.
- 公益社団法人日本薬学会の論文
- 1978-08-25
著者
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千賀 慶太郎
Pharmaceutical Institute, School of Medicine, Keio, University
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千賀 慶太郎
Pharmaceutical Institute School Of Medicine Keio University
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千賀 慶太郎
慶応大 病院
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千賀 慶太郎
慶応義塾大学病院薬剤部
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金森 由香子
Pharmaceutical Institute, School of Medicine, Keio University
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金森 由香子
Pharmaceutical Institute School Of Medicine Keio University
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西垣 貞男
慶応義塾大学病院
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