Syntheses of 9-Deazatheophyllines and 6-Deoxy-9-deazatheophyllines
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概要
- 論文の詳細を見る
The reaction of 1,3-dimethyl-5-nitro-6-styryluracils (IIa-e) with sodium dithionite in formic acid afforded the corresponding 8-aryl-9-deazatheophyllines (IVa-e). The reaction of IVa with phosphorus oxychloride gave 6-chloro-6-deoxy-8-phenyl-9-deazatheophylline (XIII), while the reaction of IVa with phosphorus oxychloride in the presence of arylamines provided the corresponding 6-arylamino-6-deoxy-8-phenyl-9-deazatheophyllines (XIV-XVI) in a single step.
- 公益社団法人日本薬学会の論文
- 1980-05-25
著者
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千賀 慶太郎
Pharmaceutical Institute, School of Medicine, Keio, University
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千賀 慶太郎
Pharmaceutical Institute School Of Medicine Keio University
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千賀 慶太郎
慶応大 病院
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千賀 慶太郎
慶応義塾大学病院薬剤部
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西垣 貞男
Pharmaceutical Institute, School of Medicine, Keio University
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金森 由香子
Pharmaceutical Institute, School of Medicine, Keio University
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金森 由香子
Pharmaceutical Institute School Of Medicine Keio University
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西垣 貞男
Pharmaceutical Institute School Of Medicine Keio University
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西垣 貞男
慶応義塾大学病院
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