THE SYNTHESIS OF 5-SUBSTITUTED 1,2,3,-TRIAZINES WITH KETENE SILYL ACETALS AND CERIC AMMONIUM NITRATE

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概要

• 論文の詳細を見る

• Monocyclic 1,2,3-triazines were reacted with ketene silyl acetal or silyl enol ether in the presence of 1-chloroethyl chloroformate to give 5-substituted 2-(1-chloroethoxycarbonyl)-2,5-dihydrotriazines. These dihydro-adducts were readily oxidized and hydrolyzed with ceric ammonium nitrate in CH_3CN/H_2O to afford 5-substituted triazines.

• 公益社団法人日本薬学会の論文
• 1995-05-15

著者

• 大沢 昭緒

  School of Pharmaceutical Sciences, Showa University

• 伊藤 喬

  昭和大学薬学部薬化学教室

• 伊藤 喬

  School of Pharmaceutical Sciences, Showa University

• 岡田 真弥子

  School of Pharmaceutical Sciences, Showa University

• 永田 和弘

  School of Pharmaceutical Sciences, Showa University

• 大沢 昭緒

  School Of Pharmaceutical Sciences Showa University

• Nagata K

  School Of Pharmaceutical Sciences Showa University

• 長谷川 博司

  School of Pharmaceutical Sciences, Showa University

• 松谷 裕二

  School of Pharmaceutical Sciences, Showa University

• 岡田 真弥子

  School Of Pharmaceutical Sciences Showa University

• 松谷 裕二

  School Of Pharmaceutical Sciences Showa University

• 長谷川 博司

  School Of Pharmaceutical Sciences Showa University

• Matsuya Y

  Graduate School Of Pharmacy And Pharmaceutical Sciences Faculty Of Pharmacy And Pharmaceutical Scien

• 永田 和弘

  School Of Pharmaceutical Sciences Showa University

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