Reaction of Six-Membered Azaaromatics with Allyltributyltin
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概要
- 論文の詳細を見る
Pyridazines were reacted with allyltributyltin in the presence of chloroformate to give 1-alkoxycarbonyl-6-allyl and 1-alkoxycarbonyl-4-allyldihydropyridazines as major and minor products, respectively. The reaction system was applied to other diazines and pyrimidine and pyrazine were shown to afford diallytetrahydroadducts. Benzodiazines also gave allylation products in good yields. The reaction seems to be applicable to most six-membered azaaromatics.
- 公益社団法人日本薬学会の論文
- 1994-09-15
著者
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大沢 昭緒
School of Pharmaceutical Sciences, Showa University
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伊藤 喬
昭和大学薬学部薬化学教室
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伊藤 喬
School of Pharmaceutical Sciences, Showa University
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岡田 真弥子
School of Pharmaceutical Sciences, Showa University
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永田 和弘
School of Pharmaceutical Sciences, Showa University
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大沢 昭緒
School Of Pharmaceutical Sciences Showa University
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Nagata K
School Of Pharmaceutical Sciences Showa University
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長谷川 博司
School of Pharmaceutical Sciences, Showa University
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松谷 裕二
School of Pharmaceutical Sciences, Showa University
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岡田 真弥子
School Of Pharmaceutical Sciences Showa University
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Hasegawa Hisashi
Sagami Research Laboratory Wakamoto Pharmaceutical Co. Ltd.
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松谷 裕二
School Of Pharmaceutical Sciences Showa University
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長谷川 博司
School Of Pharmaceutical Sciences Showa University
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Hasegawa H
Department Of Pharmaceutical Technology Kobe Pharmaceutical University
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Matsuya Y
Graduate School Of Pharmacy And Pharmaceutical Sciences Faculty Of Pharmacy And Pharmaceutical Scien
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永田 和弘
School Of Pharmaceutical Sciences Showa University
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