Reaction of 21-Bromo-17α-methoxy-20-ketopregnenes with Sodium Methoxide or Potassium Acetate

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概要

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• The reaction of 21-bromo-3β-hydroxy-17α-methoxypregn-5-en-20-one (5) with NaOCH_3 in MeOH under reflux gave the 21-aldehyde 9 in modest yield along with the 21-hydroxy derivative 6. The 21-acetates 8 and 13 were obtained in good yields by prolonged reaction of the 21-bromides 5 and 11 with CH_3COO^-.

• 公益社団法人日本薬学会の論文
• 1985-10-25

著者

• 沼沢 光輝

  Tohoku Pharmaceutical University

• 沼沢 光輝

  Tohoku College Of Pharmacy

• 長岡 正男

  東北薬科大学

• 長岡 正男

  Tohoku College of Pharmacy

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