SYNTHESIS OF (±)-FLUSTRAMINE B, A MARINE ALKALOID
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概要
- 論文の詳細を見る
6-Bromo-N_b-methoxycarbonyltryptamine (7) was prepared from 5-nitropyrroloindole (4a) by a series of reactions : reduction, bromination, deamination, and ring opening. Prenylation of 7 with an excess dimethylallyl bromide gave the 3a, 8-diprenylpyrroloindole (8). Hydrolysis of 8 followed by methylation with MeI-K_2CO_3-acetone provided (±)-flustramine B.
- 公益社団法人日本薬学会の論文
- 1983-05-25
著者
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日野 亨
Faculty of Pharmaceutical Sciences, Chiba University
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中川 昌子
千葉大薬
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日野 亨
千葉大 薬
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松木 健司
千葉大・薬
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中川 昌子
Faculty Of Pharmaceutical Sciences Hokkaido University
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中川 昌子
千葉大 薬
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田中 隆雄
Faculty of Pharmaceutical Sciences, Chiba University
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松木 健司
Faculty of Pharmaceutical Sciences, Chiba University
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田中 隆雄
Faculty Of Pharmaceutical Sciences Chiba University
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