Acylindoles. VIII. New Procedures for 1-Heteroaroylindole-3-acetic Acid Derivatives
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概要
- 論文の詳細を見る
1-Heteroaroyl-2-methylindole-3-acetic acid derivatives are prepared by reacting the corresponding N^1-heteroaroylphenylhydrazine derivatives with levulinic acid. And these indole derivatives are also prepared by some other procedures. In one of these compounds, 1-nicotinoyl-2-methyl-5-methoxyindole-3-acetic acid, the existence of its dimorph is suggested by the infrared spectrum. The indole derivatives show a remarkable experimental anti-inflammatory activity having extremely low toxicity.
- 公益社団法人日本薬学会の論文
- 1968-10-25
著者
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山本 久夫
Pharmaceuticals Divisiou, Sumitomo Chemical Co., Ltd.
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岡本 忠士
Pharmaceuticals Division Sumitomo Chemical Co. Ltd.
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山本 久夫
Research Department Pharmaceuticals Division Sumitomo Chemical Co. Ltd.
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中尾 勝
Pharmaceuticals Division, Sumitomo Chemical Co., Ltd.
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中尾 勝
Pharmaceuticals Division Sumitomo Chemical Co. Ltd.
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