Diels-Alder Reaction of 1, 3-Butadiene Derivatives with 1-Methyl-2(1H)-quinolones Having an Electron-Withdrawing Group at the 4-Position

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概要

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• Diels-Alder reactions of 1-methyl-2(1H)-quinolones having an electron-withdrawing group at the 4-position with isoprene, butadiene sulfone, and cyclohexadiene were performed to yield functionalized phenanthridones stereoselectively at atmospheric and at high pressure. Regioselectivity and stereochemistry of a methoxycarbonyl group were studied using the semi-empirical and ab initio MO methods, respectively.

• 公益社団法人日本薬学会の論文
• 2001-07-01

著者

• WATANABE Kazuhiro

  Tohoku Pharmaceutical University

• Watanabe K

  School Of Life Science Tokyo University Of Pharmacy And Life Science

• Watanabe Kazuhiro

  Tohoku Pharmaceutical Univ. Sendai Jpn

• FUJITA Reiko

  Tohoku Pharmaceutical University

• Fujita R

  Tohoku Pharmaceutical University

• Fujita R

  Department Of Chemistry School Of Liberal Arts And Sciences Iwate Medical University

• MATSUZAKI Hisao

  Tohoku Pharmaceutical University

• HONGO Hiroshi

  Tohoku Pharmaceutical University

• Hongo H

  Tohoku Pharmaceutical University

• YOSHISUJI Toshiteru

  Tohoku Pharmaceutical University

• Matsuzaki H

  Tohoku Pharmaceutical University

• Watanabe Kazuhiro

  Tohoku Natl. Agr. Exp. Stn.

• Watanabe Kazuki

  Faculty Of Pharmaceutical Sciences Aomori University

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