Total Synthesis of the Anthelmintic Cyclodepsipeptide, PF1022A
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概要
- 論文の詳細を見る
The anthelmintic cyclooctadepsipeptide PF1022A and its antipode were synthesized starting from L-N^α-Boc-leucine (for PF1022A), D-N^α-Boc-leucine (for the antipode), L-lactic acid, and L-phenyllactic acid using Mitsunobu reaction and/or the DCC/HOBt method. The antipode had no anthelmintic efficacy.
- 社団法人日本農芸化学会の論文
- 1994-06-23
著者
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Suzuki Akinori
Department Of Agricultural Chemistry Faculty Of Agriculture The University Of Tokyo
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Ohyama Makoto
Department Of Agricultural Chemistry Faculty Of Agriculture The University Of Tokyo:pharmaceutical T
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IINUMA Katsuharu
Pharmaceutical Technology Laboratories
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Iinuma Katsuharu
Pharmaceutical Technology Laboratories Meiji Seika Kaisha Ltd.
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Isogai Akira
Department Of Agricultural Chemistry Faculty Of Agriculture The University Of Tokyo
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