Total syntheses of indicine N-oxide, intermedine N-oxide, and their enantiomers using carbohydrate as a chiral educt.
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概要
- 論文の詳細を見る
The first completely enantioselective syntheses of indicine <I>N</I>-oxide, intermedine <I>N</I>-oxide, and their enantiomers have been achieved stereospecifically. A synthetic analogue modeled on indicine <I>N</I>-oxide showed the superior activity to indicine <I>N</I>-oxide itself against cancer cell in vitro test.
- 公益社団法人 日本化学会の論文
著者
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NISHIMURA Yoshio
Institute of Microbial chemistry
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KONDO Shinichi
Institute of Microbial chemistry
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Takeuchi Tomio
Institute For Chemotherapy M.c.r.f.
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Umezawa Hamao
Institute of Bioorganic Chemistry
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Nishimura Yoshio
Institute of Bioorganic Chemistry
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