Neurotropic and Psychotropic Agents. VI. 1-Alkoxymethyl-1,3-dihydro-2H-1,4-benzodiazepin-2-ones
スポンサーリンク
概要
- 論文の詳細を見る
1-Alkoxymethyl-1,3-dihydro-2H-1,4-benzodiazepin-2-ones (II) were prepared by two methods : one was direct alkylation of 1,4-benzodiazepin-2-ones (I) with alkoxymethyl chlorides and the other was via 2-[N-(alkoxymethyl) phthalimidoacetamido] benzophenones (IV) which were prepared from the corresponding 2-(phthalimidoactamido) benzophenones (III) and alkoxymethyl chlorides. Certain compounds prepared had comparable activity to diazepam and chlorodiazepoxide in taming and anticonvulsant tests in mice.
- 1982-04-25
著者
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岸本 禎二
Central Research Laboratories Fujisawa Pharmaceutical Co. Ltd.
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松尾 昌昭
New Drug Research Laboratories, Fujisawa Pharmaceutical Co., Ltd.,
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植田 育男
Central Research Laboratories Fujisawa Pharmaceutical Co. Ltd.
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松尾 昌昭
Central Research Laboratories, Fujisawa Pharmaceutical Co., Ltd.
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松尾 昌昭
New Drug Research Laboratories Fujisawa Pharmaceutical Co. Ltd.
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