Studies on 1-Alkyl-2 (1H)-pyridone Derivatives. XXII. The Friedel-Crafts Reaction of 1-Methyl-2 (1H)-pyridone and Its Homologs with Benzoyl Chloride

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概要

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• The Friedel-Crafts reaction of 1-methyl-2 (1H)-pyridone (I), 1-methyl-2 (1H)-quinolone (II), and 2-methyl-1 (2H)-isoquinolone (III) with benzoyl chloride was successfully carried out. I gave products identified as 5-benzoyl-1-methyl-2 (1H)-pyridone (IV), 3-benzoyl-1-methyl-2 (1H)-pyridone (V), and 3,5-dibenzoyl-1-methyl-2 (1H)-pyridone (VI). II gave 3-benzoyl-1-methyl-2 (1H)-quinolone (VII) and 6-benzoyl-1-methyl-2 (1H)-quinolone (VIII), and III gave 4-benzoyl-2-methyl-1 (2H)-isoquinolone (IX) and 5-benzoyl-2-methyl-1 (2H)-isoquinolone (X).

• 社団法人日本薬学会の論文
• 1974-09-25

著者

• 加藤 秀樹

  Tohoku College Of Pharmacy

• 本郷 弘司

  東北薬科大学

• 藤田 礼子

  Tohoku College of Pharmacy

• 本郷 弘司

  Tohoku College of Pharmacy

• 富沢 宏

  東北薬科大学

• 富沢 宏

  Tohoku College of Pharmacy

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