Synthesis of 1,5-Benzothiazepine Derivatives. III

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概要

• 論文の詳細を見る

• Various derivatives of 2-aryl-3-hydroxy-2,3-dihydro-1,5-benzothiazepin-4 (5H)-one (I) were synthesized. Alternative routes to 2-aryl-3-hydroxy-5-alkyl-trans-2,3-dihydro-1,5-benzothiazepin-4 (5H)-one (II-β) and 2-aryl-3-acetoxy-5-dimethylaminoethyl-cis-2,3-dihydro-1,5-benzothiazepin-4 (5H)-one (VI-α) were also investigated respectively.

• 公益社団法人日本薬学会の論文
• 1971-03-25

著者

• 井上 博純

  Organic Chemistry Research Laboratory, Tanabe Seiyaku Co., Ltd, .

• 近田 美紀彦

  Organic Chemistry Research Laboratory, Tanabe Seiyaku Co., Ltd.

• 釘田 博至

  Organic Chemistry Research Laboratory, Tanabe Seiyaku Co., Ltd.

• 竹尾 聰

  田辺製薬株式会社有機化学研究所

• 池崎 宗克

  Organic Chemistry Research Laboratory Tanabe Seiyaku Co. Ltd.

• 竹尾 聰

  Organic Chemistry Research Laboratory, Tanabe Seiyaku Co., Ltd.

• 釘田 博至

  田辺製薬有機研究所

• 釘田 博至

  Organic Chemistry Research Laboratory:tanabe Seiyaku Co. Ltd.

• 井上 博純

  Organic Chemistry Research Laboratory Tanabe Seiyaku Co. Ltd .

• 近田 美紀彦

  Organic Chemistry Research Laboratory Tanabe Seiyaku Co. Ltd.

• 釘田 博至

  Organic Chemistry Research Laboratory Tanabe Seiyaku Co. Ltd.

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