Studies on Antiatherosclerotic Agents. Synthesis of 5-Substituted Derivatives of 7-Ethoxycarbonyl-6,8-dimethyl-1(2H)-phthalazinone
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概要
- 論文の詳細を見る
Several 5-substituted derivatives of 7-ethoxycarbonyl-6,8-dimethyl-1(2H)-phthalazione were prepared by means of nitration, reductive amination, and diazonium decomposition. The substituents introduced included NO_2,NH_2,F, Cl, CN. Among the derivatives, the fluorine compound was obtained only in poor yield because intramolecular cyclization occurred predominantly.
- 公益社団法人日本薬学会の論文
- 1991-07-25
著者
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江口 征夫
Institute For Medical And Dental Engineering Tokyo Medical And Dental University
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江口 征夫
日本動脈硬化研究所
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石川 正幸
Institute For Medical And Dental Engineering Tokyo Medical And Dental University
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