A New Method for Preparing D-Penicillamine. : Reaction of Benzylpenicilloic Acid α-Amides with Arylamines
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概要
- 論文の詳細を見る
Benzylpenicilloic acid α-amides (1a-d) prepared by aminolysis of benzylpenicillin were treated with arylamines (2,7,9 and 13a-f) in the presence of acetic acid to give D-penicillamine (3) in good yield and high purity. The structures pf the by-products formed in these reactions were also determined.
- 公益社団法人日本薬学会の論文
- 1988-06-25
著者
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曽田 馨
Research Center, Taisho Pharmaceutical Co., Ltd.
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富沢 一雪
Research Center, Taisho Pharmaceutical Co., Ltd.,
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小川 利寿
Research Center, Taisho Pharmaceutical Co., Ltd.,
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冨沢 一雪
Research Center Taisho Pharmaceutical Co. Ltd.
-
小川 利寿
Research Center Taisho Pharmaceutical Co. Ltd.
-
富沢 一雪
Research Center Taisho Pharmaceutical Co. Ltd.
-
曽田 馨
Research Center Taisho Pharmaceutical Co. Ltd.
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