Synthesis of 3-Sarcosine-, 3-Glycine-, and 3-L-Alanine-6-Glycine-Bradykinin and 3-Glycine-Bradykinin.
スポンサーリンク
概要
- 論文の詳細を見る
The three analogs of bradykinin are described in which L-proline residue in 3-position of 6-glycine-bradykinin is substituted for sarcosine, glycine, and L-alanine residue respectively. 3-Glycine-bradykinin and its O-acetyl compound are also described. The biological activity of the five analogs is compared with that of bradykinin on an isolated guinea pig ileum.
- 公益社団法人日本薬学会の論文
- 1967-08-25
著者
関連論文
- Synthesis of Carboxyl-Terminal Extension Analogs of Dermorphin and Evaluation of Their Opioid Receptor-Binding and Opioid Activities
- Degradation of Deltorphins and Their Analogs by Rat Brain Synaptosomal Peptidases
- Solid-Phase Synthesis and Opioid Activities of [D-Ala^2]Deltorphin II Analogs
- Studies on Analgesic Oligopeptides. VII. Solid Phase Synthesis and Biological Properties of Tyr-D-Arg-Phe-βAla-NH_2 and Its Fluorinated Aromatic Amino Acid Derivatives
- Solid Phase Synthesis and Opioid Receptor Binding Properties of Presumable Dermorphin Precursor Derivatives
- Solid Phase Synthesis and Opioid Receptor Binding Activities of[D-Ala^2,D-Leu^5]Enkephalin Analogs Containing a Fluorinated Aromatic Amino Acid
- Studies on Analgesic Oligopeptides. VI. : Further Studies of Synthesis and Biological Properties of Tripeptide Alkylamides, Try-D-Arg-Phe-X
- Studies on analgesic Oligopeptides. V. : Structure-Activity Relationship of Tripeptide Alkylamides, Tyr-D-Arg-Phe-X
- Studies on Analgesic Oligopeptides. IV. Synthesis and Analgesic Activity of N-Terminal Shorter Analogs of [D-Arg^2] Dermorphin and Des-Tyr^1-Dermorphin Analogs
- Studies on Analgesic Oligopeptides. III. Synthesis and Analgesic Activity after Subcutaneous Administration of [D-Arg^2] dermorphin and Its N-Terminal Tetrapeptide Analogs
- Studies on Analgesic Oligopeptides. II. Structure-Activity Relationship among Thirty Analogs of a Cyclic Dipeptide, Cyclo (-Tyr-Arg-)
- Structure and Analgesic Activity Relationship of Cyclo-Tyrosyl-Arginyl and Its Three Stereoisomers
- Acetic Acid-Catalyzed Diketopiperazine Synthesis
- The β-p-Nitrobenzyl Ester to Minimize Side Reaction during Treatment of Aspartyl Peptides with Methanesulfonic Acid
- Selective Cleavage of tert-Butyloxycarbonyl Protecting Group with Dilute Organic Sulfonic Acid without Decomposition of Tryptophan Residue
- The γ-Phenacyl and γ-p-Nitrobenzyl Esters to Minimize Side Reactions during Treatment of Glutamyl Peptides with Hydrogen Fluoride-Anisole Mixture
- An Improved Attachment of N-Protected Amino Acid and Peptide to Chloromethylated Polystyrene-divinylbenzene Resin
- Tactics for Simplification of Purification Process in the Solid Phase Peptide Synthesis
- Suppression of Diketopiperazine Formation in Solid Phase Peptide Synthesis
- Synthesis of Tryptic Peptides of Hen Egg Lysozyme (Positions 1-5 and 69-73) and Related Peptides
- Synthesis of Every Kinds of Peptide Fragments of Bradykinin
- The β-Phenacyl and β-p-Nitrobenzyl Esters to Suppress Side Reactions during Treatment of Aspartyl Peptides with Hydrogen Fluoride
- Synthesis of Bradykinyl-peptide and Peptidyl-bradykinin
- Synthesis of 4-L-Valine-6-L-Threonine-, 4-L-Isoleucine-6-L-Threonine-, 4-L-Leucine-6-L-Threonine-, 4-L-Valine-, and 4-L-Isoleucinebradykinin and Their O-Acetyl Compounds.
- Synthesis of 3-Sarcosine-, 3-Glycine-, and 3-L-Alanine-6-Glycine-Bradykinin and 3-Glycine-Bradykinin.
- Synthesis of 3-L-Lysine-bradykinin and Its O-Acetyl Compound
- Synthesis of β-Alanine-containing Analogs of Bradykinin
- Synthesis of Peptides Related to the C-Therminus of B-Peptide of Ox Co-fibrin : Positions 16〜21,15〜21,and 13〜21
- Synthesis of 4-L-Leucine-6-O-acetyl-L-serine, 4-L-Leucine, 6-O-Acetyl-L-serine Bradykinin, and Bradykinin
- Synthesis of 6-L-Lecucine, 6-O-Acetyl-L-threonine, and 6-L-Threonine-bradykinin
- Studies on Encephalitogenic Fragments of Myelin Protein. IV. Synthesis of Glycine Analogs of Tryptophan-containing Fragment
- Studies on Encephalitogenic Fragments of Myelin Protein. II. Solid Phase Synthesis of Tryptophan-containing Decapeptide
- Syntheses of [Phe (4NO_2)^5,Tyr (Me)^8]-and [Tyr (Me)^5,Phe (4NO_2)^8]-Bradykinin