Synthesis of B-(sec-Amino)alanines

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概要

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• Preparation of β-(sec-amino)alanines (3) by acid hydrolysis of diethyl (sec-aminomethyl)formamidomalonates (2) was studied. Although high reaction temperature resulted in low yield, low reaction temperature (below 30℃) gave good to excellent yields. The hydrolysis of diethyl formamido(piperidinomethyl)malonate (2a) was followed by ^1H-NMR, and a plausible mechanism involving the condensation of ethyl hydrogen aminomalonate (7) with 1-piperidinemethanol (5) is proposed.

• 公益社団法人日本薬学会の論文
• 1998-01-15

著者

• SUMOTO Kunihiro

  Faculty of Pharmaceutical Sciences, Fukuoka University

• Sumoto K

  Faculty Of Pharmaceutical Sciences Fukuoka University

• Sumoto Kunihiro

  Fukuoka Univ. Fukuoka Jpn

• Sumoto Kunihiro

  Faculty Of Pharmaceutical Sciences Fukuoka University

• FUJISAKI Fumiko

  Faculty of Pharmaceutical Sciences, Fukuoka University

• ABE Nobuhiro

  Faculty of Pharmaceutical Sciences, Fukuoka University

• Fujisaki Fumiko

  Faculty Of Pharmaceutical Sciences Fukuoka University

• Sumoto Kunihiro

  Faculty of Pharmaceutical Science, Fukuoka University

• Fujisaki Fumiko

  Faculty of Pharmaceutical Science, Fukuoka University

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