Effective Synthesis of Optically Active Trifluoromethyldiazirinyl Homophenylalanine and Aroylalanine Derivatives with the Friedel-Crafts Reaction in Triflic Acid

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概要

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• The Friedel-Crafts reaction with 3-(3-methoxyphenyl)-3-(trifluoromethyl)-3H-diazirine and optically active N-TFA-Asp(Cl)-OMe in triflic acid afforded homophenylalanine derivatives without any loss of the optical purity.

• 社団法人 日本農芸化学会の論文
• 2009-06-23

著者

• 橋本 誠

  北海道大学大学院農学研究院

• HASHIMOTO Makoto

  Department of Dermatology, Asahikawa Medical College

• Hatanaka Yasumaru

  Graduate School Of Medicine And Pharmaceutical Sciences University Of Toyama

• Hatanaka Yasumaru

  Fac. Of Pharmaceutical Sciences Toyama Medical And Pharmaceutical Univ.

• Hashimoto Makoto

  Department Of Dermatology Asahikawa Medical College

• Hashimoto Makoto

  Obihiro Univ. Agriculture And Veterinary Medicine Hokkaido Jpn

• MURASHIGE Ryo

  Department of Agricultural and Life Science, Obihiro University of Agriculture and Veterinary Medici

• MURAI Yuta

  Department of Agricultural and Life Science, Obihiro University of Agriculture and Veterinary Medici

• Hashimoto Makoto

  Div. Of Applied Sci. Graduate School Of Agriculture Hokkaido Univ.

• MURAI Yuta

  Division of Applied Science, Graduate School of Agriculture, Hokkaido University

• Hashimoto Makoto

  Department Of Agricultural And Life Science Obihiro University Of Agriculture And Veterinary Medicin

• Hashimoto Makoto

  Department Of Agricultural And Life Science Obihiro University Of Agriculture And Veterinary Medicin

• Hashimoto Makoto

  Department Of Bioresource Science Obihiro University Agriculture

• Hashimoto Makoto

  Department Of Biology And Biochemistry University Of Bath:department Of Bioresource Science Obihiro

• Hashimoto Makoto

  Department Of Agricultural And Life Science Obihiro University Of Agriculture And Veterinary Medicin

• Murai Yuta

  Div. Of Applied Sci. Graduate School Of Agriculture Hokkaido Univ.

• Hatanaka Yasumaru

  Graduate School Of Medicine And Pharmaceutical Science University Of Toyama

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