Characteristics of Inhibitory Effects of Serotonin (5-HT)_3 - Receptor Antagonists, YM060 and YM114 (KAE - 393), on the von Bezold - Jarisch Reflex Induced by 2 - Methyl - 5 - HT, Veratridine and Electrical Stimulation of Vagus Nerves in Anesthetized Rats
スポンサーリンク
概要
- 論文の詳細を見る
- 1995-12-01
著者
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Miyata K
Yamanouchi Pharmaceutical Co. Ltd. Ibaraki Jpn
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Miyata K
Yamanouchi Pharmaceutical Co. Ltd. Tsukuba City Jpn
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Miyata Keiji
Inflammation Research Pharmacology Laboratories Institute For Drug Discovery Research Yamanouchi Pha
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Miyata Keiji
Neuroscience/gastrointestinal Research Laboratories Institute For Drug Discovery Research Yamanouchi
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Miyata Keiji
Neuroscience And Gastrointestinal Research Laboratory Institute For Drug Discovery Research Yamanouc
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Miyata K
Institute For Drug Discovery Research Yamanouchi Pharmaceutical Co.
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Koide T
Hiroshima Univ. Higashi‐hiroshima‐shi Jpn
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YAMANO Mayumi
Neuroscience and Gastrointestinal Research Laboratories, Institute for Drug Discovery Research, Yama
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KAMATO Takeshi
Neuroscience and Gastrointestinal Research Laboratories, Institute for Drug Discovery Research, Yama
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ITO Hiroyuki
Neuroscience Research, Pharmacology Laboratories, Institute for Drug Discovery Research, Yamanouchi
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Yamano Mayumi
Pharmacology Laboratories Institute For Drug Discovery Research Yamanouchi Pharmaceutical Co. Ltd.
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Miyata K
Inflammation Research Pharmacology Laboratories Institute For Drug Discovery Research Yamanouchi Pha
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Miyata K
Hitachi Research Laboratory Hitachi Ltd.
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Yamano Mayumi
Neuroscience And Gastrointestinal Research Laboratories Institute For Drug Discovery Research Yamano
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Ito Hiroyuki
Pharmacology Laboratories Institute For Drug Discovery Research Yamanouchi Pharmaceutical Co. Ltd.
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Ito Hiroyuki
Neuroscience And Gastrointestinal Research Laboratory Institute For Drug Discovery Research Yamanouc
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Kamato Takeshi
Neuroscience & Gastrointestinal Research Laboratories, Institute for Drug Discovery Research, Yamanouchi Pharmaceutical Co., Ltd.
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Yamano Mayumi
Neuroscience & Gastrointestinal Research Laboratory, Institute for Drug Discovery Research, Yamanouchi Pharmaceutical Co., Ltd.
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Miyata Keiji
Neuroscience & Gastrointestinal Research Laboratories, Institute for Drug Discovery Research, Yamanouchi Pharmaceutical Co., Ltd.
関連論文
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- Biological Activity of Analogues of YM022. Novel (3-Amino Substituted Phenyl)urea Derivatives of 1,4-Benzodiazepin-2-one as Gastrin : Cholecystokinin-B Receptor Antagonists
- In Vivo Pharmacologic Profile of YM158, a New Dual Antagonist for Leukotriene D_4 and Thromboxane A_2 Receptors
- Effect of YM158, a Dual Lipid Mediator Antagonist, on Immediate and Late Asthmatic Responses, and on Airway Hyper-responsiveness in Guinea Pigs
- Effect of Serotonin (5 - HT)_3 - Receptor Antagonists YM060, YM114 (KAE - 393), Ondasetron and Granisetron on 5 - HT_4 Receptors and Gastric Emptying in Rodents
- Comparative Study of [^3H]Ramosetron and [^3H]Granisetron Binding in the Cloned Human 5 : Hydroxytryptamine_3 Receptors
- The Selective 5 : Hydroxytryptamine (5 : HT)_4 : Receptor Agonist RS67506 Enhances Lower Intestinal Propulsion in Mice
- Protective Effect of a Pancreatic Elastase Inhibitor Against a Variety of Acute Pancreatitis in Rats
- Pancreatic Enzyme-Induced Pancreatitis and Systemic Complications in Rats
- Species Differences in the 5-Hydroxytryptamine-Induced Contraction in the Isolated Distal Ileum
- Characteristics of Inhibitory Effects of Serotonin (5-HT)_3 - Receptor Antagonists, YM060 and YM114 (KAE - 393), on the von Bezold - Jarisch Reflex Induced by 2 - Methyl - 5 - HT, Veratridine and Electrical Stimulation of Vagus Nerves in Anesthetized Rats
- Studies on Serotonin (5-HT)_3-Receptor Antagonist Effects of Enantiomers of 4,5,6,7-Tetrahydro-1H-Benzimidazole Derivatives
- YM-40461 Improves Airway Clearance in Guinea Pigs with Induced Subacute Bronchitis
- YM-40461, a Potent Surfactant Secretagogue, Improves Mucocilliary Clearance in SO_2-Exposed Guinea Pigs
- Synthesis of the Selective 5-Hydroxytryptamine 4 (5-HT_4) Receptor Agonist (+)-(S)-2-Chloro-5-methoxy-4-[5-(2-piperidylmethyl)-1,2,4-oxadiazol-3-yl]aniline
- Novel 5-Hydroxytryptamine 4 (5-HT_4) Receptor Agonists. Synthesis and Gastroprokinetic Activity of 4-Amino-N-[2-(1-aminocycloalkan-1-yl)ethyl]-5-chloro-2-methoxybenzamides
- Novel 5-Hydroxytryptamine (5-HT_3) Receptor Antagonists. Synthesis and Structure-Activity Relationships of 9-Methyl-2,3,4,9-tetrahydrothiopyrano[2,3-b]indol-4-one Derivatives
- Novel 5-Hydroxytryptamine (5-HT_3) Receptor Antagonists. IV. Synthesis and Pharmacological Evaluation of the Oxidation Products of (-)-(R)-5-[(1-Methyl-1H-indol-3-yl)carbonyl]-4,5,6,7-tetrahydro-1H-benzimidazole Hydrochloride (YM060 : Ramosetron)
- Novel 5-Hydroxytryptamine (5-HT_3) Receptor Antagonists. III. Pharmacological Evaluations and Molecular Modeling Studies of Optically Active 4,5,6,7-Tetrahydro-1H-benzimidazole Derivatives
- Novel 5-Hydroxytryptamine (5-HT_3) Receptor Antagonists. II. Synthesis and Structure-Activity Relationships of 4,5,6,7-Tetrahydro-1H-benzimidazole Derivatives
- Novel 5-Hydroxytryptamine (5-HT_3) Receptor Antagonists. I. Synthesis and Structure-Activity Relationships of Conformationally Restricted Fused Imidazole Derivatives
- Antisecretory and Antiulcer Effects of YM020, a New H^+, K^+-ATPase Inhibitor, in Rats and Dogs
- Comparative Evaluation of the Role of Endogenous Gastrin in Basal Acid Secretion in Conscious Rats Provided with Chronic Fistula and Pylorus Ligation
- YM-231146, a Novel Orally Bioavailable Inhibitor of Vascular Endothelial Growth Factor Receptor-2, Is Effective against Paclitaxel Resistant Tumors(Pharmacology)
- Leakage Current Reduction of Poly-Si Thin Film Transistors by Two-Step Annealing
- Mixed Planar and H-V Over-the-Cell Routing for Standard Cells with Nonuniform Over-the-Cell Routing Capacities (Special Issue on Synthesis and Verification of Hardware Design)
- An Efficient Timing-Driven Global Routing Method for Standard Cell Layout (Special Issue on Synthesis and Verification of Hardware Design)
- A Floorplanning Method with Topological Constraint Manipulation in VLSI Building Block Layout (Special Section on VLSI Design and CAD Algorithms)
- A Graph Bisection Algorithm Based on Subgraph Migration (Special Section on VLSI Design and CAD Algorithms)
- An Optimal Channel Pin Assignment Algorithm for Hierarchical Building-Block Layout Design (Special Section on VLSI Design and CAD Algorithms)
- Large-Area Doping Process for Fabrication of poly-Si Thin Film Transistors Using Bucket Ion Source and XeCl Excimer Laser Annealing
- TEM Observations of Initial Crystallization States for LPCVD Si Films : Condensed Matter
- Histamine H2-Receptor Plays Only a Minor Role in Histamine-Induced Wheal Response in the Squirrel Monkey and Guinea Pig.
- Antisecretory Effects of a Novel and Long-Lasting Histamine H2-ReceptorAntagonist, YM-14471, in Rats and Dogs.
- Serotonin (5-HT)3-Receptor Antagonism of 4,5,6,7-Tetrahydrobenzimidazole Derivatives against 5-HT-Induced Bradycardia in Anesthetized Rats.