Zinc Triflate-Promoted Glycosidation : Synthesis of Lipid A Disaccharide Intermediates
スポンサーリンク
概要
- 論文の詳細を見る
Zinc triflate was found to be superior to the heavy metal salts as a promoter in the Koenigs-Knorr type glycosidation reaction in the synthesis of lipid A disaccharide intermediates. It readily promoted the reaction of a complex glycosyl bromide with a reducing sugar moiety and gave the disaccharide with β-selectivity in good yield. This method would be suitable for the bulk preparation of lipid A disaccharide intermediates.
- 社団法人日本薬学会の論文
- 1992-11-25
著者
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東 邦雄
Drug Delivery System Institute Ltd.
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日馬 恒雄
Exploratory Research Laboratories I Daiichi Pharmaceutical Co. Ltd.
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中山 清
Exploratory Research Laboratories I, Daiichi Pharmaceutical Co. Ltd.,
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東 邦雄
Exploratory Research Laboratories I, Daiichi Pharmaceutical Co. Ltd.,
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曽我 恒彦
Exploratory Research Laboratories I, Daiichi Pharmaceutical Co. Ltd.,
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魚戸 浩一
Exploratory Research Laboratories I, Daiichi Pharmaceutical Co. Ltd.,
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中山 清
Exploratory Research Laboratories I Daiichi Pharmaceutical Co. Ltd.
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魚戸 浩一
Exploratory Research Laboratories I Daiichi Pharmaceutical Co. Ltd.
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曽我 恒彦
Exploratory Research Laboratories I Daiichi Pharmaceutical Co. Ltd.
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