Bischler-Napieralski Reactions of N-(2-Indolylethyl) acetamide
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概要
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Bischler-Napieralski reaction of N-(2-indol-4-ylethyl) acetamide (II) gave pyridoindole (III) and azepinoindole (IV), N-(2-indol-5-ylethyl) acetamide (V) afforded pyridoindoles (VI and VII), N-(2-indol-6-ylethyl) acetamide (XIII) gave pyridoindoles (XIII and XIV) and N-(2-indol-7-ylethyl) acetamide (XIX) yielded pyridoindole (XX). These reactivity of indole was supported by calculated charge density with CNDO/2.
- 公益社団法人日本薬学会の論文
- 1975-12-25
著者
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寺田 敦祐
Central Research Laboratories, Sankyo Co., Ltd.
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寺田 敦祐
京都薬科大学 化学研究所
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成戸 俊二
Central Research Laboratories, Sankyo Co.
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成戸 俊二
New Lead Research Laboratories
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Terada A
Medicinal Chemistry Research Laboratories Sankyo Co. Ltd.
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