Formation of Triazole and Isoxazole Derivatives from β-Substituted Pyridinium Salts
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概要
- 論文の詳細を見る
Treatment of 1-methyl-3-(3-phenyl-1-triazenyl) pyridinium iodide (2a-e) with base gave triazole derivatives (3 and 4) with expulsion of the pyridine ring. Similarly, the reaction of 1-methyl-3-benzoylpyridinium oxime iodide (10a-c) with base afforded isoxazole derivatives. A possible mechanism for the formation of these reaction products is discussed.
- 公益社団法人日本薬学会の論文
- 1980-07-25
著者
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田中 茂
Central Research Laboratories Sankyo Co. Ltd.
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寺田 敦祐
Central Research Laboratories, Sankyo Co., Ltd.
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和智 一之
京都薬科大学 化学研究所
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寺田 敦祐
京都薬科大学 化学研究所
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和智 一之
Central Research Laboratories, Sankyo Co., Ltd.
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Terada A
Medicinal Chemistry Research Laboratories Sankyo Co. Ltd.
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