Unexpected Catalytic Behavior of Chiral Bisoxazoline in Asymmetric Reaction of Lithium Ester Enolate with Imine
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概要
- 論文の詳細を見る
Reaction of a lithium ester enolate with benzaldehyde anisidine-imine was catalyzed by a catalytic amount of bisoxazoline ligand to afford the corresponding β-lactam in higher ee than that obtained by the reaction using a stoichiometric amount of the ligand. Investigation of the varying factors suggested the involvement of steric factors.
- 公益社団法人日本薬学会の論文
- 1999-05-15
著者
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TOMIOKA Kiyoshi
Graduate School of Pharmaceutical Sciences, Kyoto University
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Tomioka Kiyoshi
Graduate School Of Pharmaceutical Sciences Kyoto Univ.
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Kambara Takeshi
Graduate School Of Pharmaceutical Sciences Kyoto University
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Kambara Takeshi
Graduate School of Information Systems, University of Electro-Communications:Department of Applied Physics and Chemistry, University of Electro-Communications
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