New Entry of Coupling Reaction of Phenacylamine Derivatives with Silylstannane

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概要

• 論文の詳細を見る

• The new coupling reaction of phenacylamines with silylstannane and lithium diisopropylamide (LDA) is reported. The treatment of a phenacylamine iodide 1 with (trimethylsilyl)tributylstannane (Me_3SiSnBu_3) and cesium fluoride (CsF) gave a dimerization product 2 having no iodine atom. Reaction of 1 with LDA afforded a dimerization product 3 with an iodine atom. The products 2 and 3 were separated to the meso and racemic isomers, respectively.

• 公益社団法人日本薬学会の論文
• 2002-03-01

著者

• Yamauchi Aiko

  Fac. Of Pharmaceutical Sciences The Univ. Of Tokushima

• Yamauchi Aiko

  Graduate School Of Pharmaceutical Sciences The University Of Tokushima

• KIHARA Masaru

  Graduate School of Pharmaceutical Sciences, The University of Tokushima

• 岩井 雄二

  Faculty Of Pharmaceutical Sciences Kobe Gakuin University

• Yamauchi A

  Fac. Of Pharmaceutical Sciences The Univ. Of Tokushima

• Iwai Y

  Kitasato Institute For Life Sciences Kitasato University

• Yamauchi A

  Graduate School Of Bioagricultural Science Nagoya University

• Kihara M

  Graduate School Of Pharmaceutical Sciences The University Of Tokushima

• IWAI Yasumasa

  Graduate School of Pharmaceutical Sciences, The University of Tokushima

• KITA Kumiko

  Graduate School of Pharmaceutical Sciences, The University of Tokushima

• MATSUSHITA Yoko

  Graduate School of Pharmaceutical Sciences, The University of Tokushima

• Kita K

  Graduate School Of Pharmaceutical Sciences The University Of Tokushima

• Matsushita Yoko

  Graduate School Of Pharmaceutical Sciences The University Of Tokushima

• Kita Kumiko

  Graduate School Of Pharmaceutical Sciences The University Of Tokushima

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