New Entry of Coupling Reaction of Phenacylamine Derivatives with Silylstannane
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概要
- 論文の詳細を見る
The new coupling reaction of phenacylamines with silylstannane and lithium diisopropylamide (LDA) is reported. The treatment of a phenacylamine iodide 1 with (trimethylsilyl)tributylstannane (Me_3SiSnBu_3) and cesium fluoride (CsF) gave a dimerization product 2 having no iodine atom. Reaction of 1 with LDA afforded a dimerization product 3 with an iodine atom. The products 2 and 3 were separated to the meso and racemic isomers, respectively.
- 公益社団法人日本薬学会の論文
- 2002-03-01
著者
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Yamauchi Aiko
Fac. Of Pharmaceutical Sciences The Univ. Of Tokushima
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Yamauchi Aiko
Graduate School Of Pharmaceutical Sciences The University Of Tokushima
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KIHARA Masaru
Graduate School of Pharmaceutical Sciences, The University of Tokushima
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岩井 雄二
Faculty Of Pharmaceutical Sciences Kobe Gakuin University
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Yamauchi A
Fac. Of Pharmaceutical Sciences The Univ. Of Tokushima
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Iwai Y
Kitasato Institute For Life Sciences Kitasato University
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Yamauchi A
Graduate School Of Bioagricultural Science Nagoya University
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Kihara M
Graduate School Of Pharmaceutical Sciences The University Of Tokushima
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IWAI Yasumasa
Graduate School of Pharmaceutical Sciences, The University of Tokushima
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KITA Kumiko
Graduate School of Pharmaceutical Sciences, The University of Tokushima
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MATSUSHITA Yoko
Graduate School of Pharmaceutical Sciences, The University of Tokushima
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Kita K
Graduate School Of Pharmaceutical Sciences The University Of Tokushima
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Matsushita Yoko
Graduate School Of Pharmaceutical Sciences The University Of Tokushima
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Kita Kumiko
Graduate School Of Pharmaceutical Sciences The University Of Tokushima
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