Synthesis of (±)-trans- or cis-(5-Aminomethyltetrahydrofuranyl)imidazole by Mitsunobu Cyclization : Synthetic Studies toward Novel Histamine H_3 or H_4-Ligands

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he (±)-trans- or cis-4(5)-(5-aminomethyltetrahydrofurany)imidazole [1 and 2| were synthesized by the Mitsunobu cyclization, starting from L-glutamic acid.
公益社団法人日本薬学会の論文
2003-03-01

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