Larvicidal Activity of (-)-Dihydroguaiaretic Acid Derivatives against Culex pipiens
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概要
- 論文の詳細を見る
The larvicidal activity against Culex pipiens of all stereoisomers of dihydroguaiaretic acid (DGA) and secoisolariciresinol was measured, and these DGAs were found to be potent. Sixteen (−)-DGA derivatives were then newly synthesized to analyze their structure-activity relationship. Two derivatives monohydroxylated at the 3- or 4-position of the 7-phenyl group of DGA induced acute paralytic activity in the mosquitoes. Derivatives with several hydroxyl groups had lower activity than the natural compound, suggesting that hydrophobicity was probably an important factor for their insecticidal activity.
- 社団法人 日本農芸化学会の論文
- 2011-09-23
著者
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YAMAUCHI Satoshi
Faculty of Agriculture, Ehime University
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Akamatsu Miki
Graduate School Of Agriculture Kyoto University
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Shuto Yoshihiro
Faculty Of Agriculture Ehime University
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Nishiwaki Hisashi
Faculty Of Agriculture Ehime University
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Yamauchi Satoshi
Faculty Of Agriculture Ehime University
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KAWAGUCHI Yuya
Faculty of Agriculture, Ehime University
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HASEBE Ayaka
Faculty of Agriculture, Ehime University
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Yamauchi Satoshi
Fac. Of Agriculture Ehime Univ.
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Hasebe Ayaka
Faculty Of Agriculture Ehime University
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Kawaguchi Yuya
Faculty Of Agriculture Ehime University
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