Stereoselective Synthesis of Tetrahydronaphthocyclobuta[1,2-d]pyrimidinediones from 5-Fluoro-1,3-dimethyluracil and Naphthalenes

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概要

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• Upon UV-irradiation in the presence of piperylene, 5-fluoro-1,3-dimethyluracil (5-FDMU) couples with naphthalenes having either an electron-withdrawing group or an electron-donating group by way of 1,2-cycloaddition via mode selectivity to give the corresponding naphthocyclobutapyrimidines regio- and stereo-selectively.

• 公益社団法人日本薬学会の論文
• 2005-02-01

著者

• Seki K

  Central Institute Of Isotope Science (graduate School Of Medicine) Hokkaido University

• Seki Koh-ichi

  Central Institute Of Isotope Science Hokkaido University

• OHKURA Kazue

  Faculty of Pharmaceutical Sciences, Health Sciences University of Hokkaido

• Ohkura Kazue

  Faculty Of Pharmaceutical Sciences Health Sciences University Of Hokkaido

• Ohkura Kazuto

  Department Of Biological Science And Technology Faculty Of Engineering The University Of Tokushima

• Ohkura Kazuto

  Department Of Applied Biological Sciences School Of Agricultural Sciences Nagoya University

• ISHIHARA Tetsuya

  Faculty of Pharmaceutical Sciences, Health Sciences University of Hokkaido

• NISHIJIMA Ken-ichi

  Faculty of Pharmaceutical Sciences, Health Sciences University of Hokkaido

• DIAKUR James

  Faculty of Pharmacy & Pharmaceutical Sciences, University of Alberta

• Ohno Kosei

  Faculty Of Pharmaceutical Sciences Health Sciences University Of Hokkaido

• Okazaki K

  Faculty Of Human Life Science Shikoku University

• Diakur James

  Faculty Of Pharmacy & Pharmaceutical Sciences University Of Alberta

• Seki Koh-ichi

  Central Institute Of Isotope Science (graduate School Of Medicine) Hokkaido University

• OHKURA Kazue

  Faculty of Phamaceutical Science, Health Sciences University of Hokkaido

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