A SIMPLE SYNTHESIS OF THE INDOLE ALKALOID BIPOLARAMIDE AND ITS DERIVATIVES
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概要
- 論文の詳細を見る
The first total synthesis of bipolaramide was achieved in 47% overall yield from (2S__-)-2,3-dihydroindole-2-carboxylic acid in three steps, utilizing thallium chemistry. Some derivatives, with dihalogeno or dialkenyl substituents at the 4 and 11 positions of (6aS__--cis)-6a, 7,13a, 14-tetrahydropyrazino[1,2-a : 4,5-a']diindole-6,13-dione have also prepared.
- 1989-12-25
著者
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染井 正徳
Faculty of Parmaceutical Sciences, Kanazawa University
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川崎 俊哉
Faculty of Pharmaceutical Sciences, Kanazawa University
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川崎 俊哉
Faculty Of Pharmaceutical Sciences Kanazawa University
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