BORONATION-THALLATION, A NEW APPROACH TO THE SYNTHESIS OF INDOLES HAVING ARYL AND/OR A HETEROARYL SUBSTITUENT AT THE 4-POSITION
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概要
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A new coupling reaction for unsymmetrical biaryls was developed and applied successfully to the syntheses of 4-arylindoles. Photoreaction of 4-halogenoindoles also proved to be a useful method for preparing 4-substituted indoles. An alternative method for synthesizing 4-(3-pyridyl)-3-indolecarbaldehyde is also reported.
- 1986-09-25
著者
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染井 正徳
Faculty of Parmaceutical Sciences, Kanazawa University
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甘利 裕邦
Faculty Of Pharmaceutical Sciences Kanazawa University
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巻田 吉彦
Faculty Of Phermaceutical Sciences Kanazawa University
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巻田 吉彦
Faculty Of Pharmaceutical Sciences Kanazawa University
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