ACRIDONES FROM THE REACTION OF N-LITHIO ANTHRANILATES WITH BENZYNES. A SHORT SYNTHESIS OF ACRONYCINE
スポンサーリンク
概要
- 論文の詳細を見る
The lithium salt of methyl N-methylanthranilate reacted with the benzyne derived in situ from aryl halides to give a N-methylacridone derivatives in a one-pot process. Using this method, a short synthesis of acronycine has been achieved.
- 公益社団法人日本薬学会の論文
- 1984-03-25
著者
-
古川 淳
Faculty of Pharmaceutical Sciences, Nagasaki University
-
渡辺 三明
Faculty of Pharmaceutical Sciences
-
渡辺 三明
Center For Instrumental Analysis Nagasaki University
-
黒崎 亜紀夫
Faculty of Pharmaceutical Sciences, Nagasaki University
-
黒崎 亜紀夫
Faculty Of Pharmaceutical Sciences Nagasaki University
関連論文
- Stable Sulfur Ylides. XII. : Reaction of 3-Alkyl(aryl)thio-silyloxydienes Derived from Stable Sulfur Ylides with Aromatic Aldehydes. : Synthesis and Structure of Thiolanium Ylides
- An Efficient Synthesis of Phthalides by Diels-Alder Reaction of Sulfur-Substituted Furanones with Silyloxydienes : A Formal Synthesis of Mycophenolic Acid
- An Efficient Synthesis of 2(5H)-Furanone and Furan Derivatives Using 3-(Phenylthio)propenal as a 1,3-Dipolar Synthon
- A Regioselective Lithiation of ortho-Cresols Using the Bis(dimethylamino)phosphoryl Group as a Directing Group : General Synthesis of 2,3-Dihydrobenzo[b]furans Including Naturally Occurring Neolignans
- A Short and Convergent Synthesis of the Phytoalexins Vignafuran, 6-Demethylvigafuran, and Moracin M via Directed Lithiation Reaction
- A Facile Synthesis of Benzo[b]furan Derivatives Including Naturally Occurring Neolignans via Regioselective Lithiation of ortho-Cresols Using the Bis(dimethylamino)phosphoryl Group as a Directing Group
- The Directed ortho-Lithiation of Aryl Tetramethylphosphorodiamidates
- Correlations between Carbon-13 Nuclear Magnetic Resonance Chemical Shifts and Reactivities of Siloxybutadienes and Siloxyazabutadienes in the Diels-Alder Reaction with Dimethyl Acetylenedicarboxylate
- Reactions of Lithiated ortho-Toluamides and Related Compounds with Vinylsilanes : Syntheses of 1-Tetralones and 1-Naphthols
- Stable Sulfur Ylides. X. : Reactions of Carbonyl-Stabilized Sulfonium Ylides with Acetyl Chloride
- Stable Sulfur Ylides. XI. : Facile Preparation of Silyloxydienes from Stable Sulfur Ylides
- LITHIATION OF ORTHO-TOLYL TETRAMETHYLPHOSPHORODIAMIDATES : A FACILE SYNTHESIS OF 2-ARYLBENZOFURANS INCLUDING NEOLIGNAN, CARINATIN
- ORTHO-LITHIATION OF PHENOLS USING THE BIS(DIMETHYLAMINO)PHOSPHORYL GROUP AS A DIRECTING GROUP
- Ring Clreavage Reaction of 1,3-Oxazine-2,4(3H)-dione Derivatives with Amines
- Total Synthesis of the Antibiotic WS-5995A Using a Key Reaction of o-Toluamide Anions with Homophthalic Anhydrides
- Regioselective Syntheses of Substituted Thioxanthen- and Selenoxanthen-9-one Derivatives
- Primidine Derivatives. V. : Synthesis and Nucleophilic Reactions of 5-Bromo-6-bromomethyl-1-(2-bromoethyl and 2-bromopropyl)-3-methyl-2,4(1H, 3H)-pyrimidinedione
- Synthesis and Reactions of 2,3-Dihydrothiazolo[3,2-α]pyrimidine Derivatives(Organic,Chemical)
- Synthesis of 5,5'-Mehylenebispyrimidine Derivatives and 3,4-Dithia[6.1](1.5)pyrimidinophane
- 安定イオウイリドの研究(第9報)Dimethylsulfonium AcetylcarbamoylmethylideとIsoquinoline 2-Oxideとの反応
- Stable Sulfur Ylides. VIII. The Reactions of 1,3-Oxazin-4-one Derivatives
- Stable Sulfur Ylides. VII. The Reaction of Dimethylsulfonium Acetylcarbamoylmethylide with Quinoline 1-Oxide
- Triphenylphosphonium Allylide類と塩基との反応
- 安定イオウイリドの研究(第6報)Dimethylsulfonium AcetylmethoxycarbonylmethylideおよびDimethylsulfonium DiacetylmethylideとIsoquinoline 2-Oxideとの反応
- Stable Sulfur Ylides. V. Syntheses of α-Acylfuran Derivatives by Thermal and Photochemical Reaction of Allylides
- Stable Sulfur Ylides. IV. Reaction of Dimethylsulfonium Acetylmethoxycarbonylmethylide and Dimethylsulfonium Diacetylmethylide with Quinoline 1-Oxide
- Stable Sulfur Ylides. III. Reaction of Stable Sulfonium Allylides and Oxosulfonium Allylides with Alkoxides
- Stable Sulfur Ylides. II. : Syntheses of Stable Sulfonium Allylides and Oxosulfonium Allylides
- Directed Lithiation反応を利用するAnthraquinone類の合成
- An Annulation Reaction to Naphthalene-1,4-diols Using Dimethyl Phthalide-3-phosphonates
- Reaction of Lithiated Senecioamide and Related Compounds with Benzynes : Efficient Syntheses of Naphthols and Naphthoquinones
- 長所をのばし定着化を(ポスターセッションの問題点を探ぐる)
- ACRIDONES FROM THE REACTION OF N-LITHIO ANTHRANILATES WITH BENZYNES. A SHORT SYNTHESIS OF ACRONYCINE
- A Regiospecific Synthesis of Anthracyclinones Using Directed Metalation
- 「1次文献」重視で主体性の確立を(情報洪水にいかに対処するか)
- 芳香環の “Directed Metalation” 反応を利用した有機合成
- 安定イオウイリドの研究(第1報)Dimethyloxo-およびDimethylsulfonium BenzoylmethylideとAromatic Amine N-Oxide類との反応
- Benzofuro[2,3-c]pyridazine誘導体の合成
- Thianaphtheno[2,3-c]pyridazine誘導体の合成