Synthesis of 2, 3-Disubstituted Indole Using Palladium(II)-Catalyzed Cyclization with Alkenylation Reaction

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概要

• 論文の詳細を見る

• The reaction of ehyl 2-ethynylphenylcarbamate derivative with alkenes in the presence of a palladium(II)catalyst, copper dichloride and tetrabutylammonium fluoride(TBAF)produced 2-substituted 3-ethenylinodoles during refluxing. The intramolecular cyclization reaction of ethyl 2-ethynylphenylcarbamates, which have an ethenyl part in the ethynyl group, was also used to produce carbazole derivatives.

• 公益社団法人日本薬学会の論文
• 2002-02-01

著者

• SAKAMOTO Takao

  Graduate School of Pharmaceutical Sciences, Tohoku University

• Suzuki N

  Graduate School Of Pharmaceutical Sciences Tohoku University

• SUZUKI Naoyuki

  Graduate School of Pharmaceutical Sciences, Tohoku University

• YASUHARA Akito

  Graduate School of Pharmaceutical Sciences, Tohoku University

• TAKEDA Yousuke

  Graduate School of Pharmaceutical Sciences, Tohoku University

• Takeda Yousuke

  Graduate School Of Pharmaceutical Sciences Tohoku University

• Yasuhara A

  Graduate School Of Pharmaceutical Sciences Tohoku University

• Yasuhara Akito

  Faculty Of Pharmaceutical Sciences Tohoku University

• Sakamoto Takao

  Graduate School Of Pharmaceutical Sciences Tohoku University

• Sakamoto T

  Second Department Of Surgery Toyama Medical And Pharmaceutical University

• Sakamoto T

  School Of Pharmacy Tokyo University Of Pharmacy And Life Science

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