Convenient Indole Synthesis from 2-Iodoanilines and Terminal Alkynes by the Sequential Sonogashira Reaction and the Cyclization Reaction Promoted by Tetrabutylammonium Fluoride (TBAF)

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概要

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• The sequential Sonogashira reaction and the cyclization reaction of various 2-iodoanilines and terminal alkynes in the presence of a palladium catalyst and tetrabutylammonium fluoride (TBAF) gave the corresponding 2-substituted indoles in good yields.

• 公益社団法人日本薬学会の論文
• 2003-10-01

著者

• SAKAMOTO Takao

  Graduate School of Pharmaceutical Sciences, Tohoku University

• Suzuki N

  Graduate School Of Pharmaceutical Sciences Tohoku University

• SUZUKI Naoyuki

  Graduate School of Pharmaceutical Sciences, Tohoku University

• YASAKI Sakura

  Graduate School of Pharmaceutical Sciences, Tohoku University

• YASUHARA Akito

  Graduate School of Pharmaceutical Sciences, Tohoku University

• Yasaki Sakura

  Graduate School Of Pharmaceutical Sciences Tohoku University

• Yasuhara A

  Graduate School Of Pharmaceutical Sciences Tohoku University

• Yasuhara Akito

  Faculty Of Pharmaceutical Sciences Tohoku University

• Sakamoto Takao

  Graduate School Of Pharmaceutical Sciences Tohoku University

• Sakamoto T

  Second Department Of Surgery Toyama Medical And Pharmaceutical University

• Sakamoto T

  School Of Pharmacy Tokyo University Of Pharmacy And Life Science

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