A NEW STABLE PROSTACYCLIN ANALOGUE OP41483 : 15-CYCLOPENTYL-ω-PENTANOR-5(E)-CARBACYCLIN
スポンサーリンク
概要
- 論文の詳細を見る
Effects of a new stable prostacyclin analogue OP41483 (15-cyclopentyl-ω-pentanor-5(E)-carbacyclin) on platelet aggregation ,plasma thromboxane B_2 levels, hemodynamic parameters, and clinical safety were studied. Normal volunteers received intravenous infusions of OP41483 at doses of 2.5 (n=3), 5.0 (n=3), 10 (n=3), and 20 (n=5) ng/kg/min for one hour. During infusion, ADP (adenosine diphosphate)-induced platelet aggregation decreased significantly, and blood pressure decreased slightly, but plasma thromboxane B_2 levels did not change significantly. The intravenous infusion of OP41483 at the dose of 10 ng/kg/min for one hour over three successive days was performed. During the each infusion, platelet aggregation and mean blood pressure decresed significantly.
- 社団法人日本循環器学会の論文
- 1985-06-20
著者
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Yui Yoshiki
Third Division Department Of Internal Medicine Faculty Of Medicine Kyoto University
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Takatsu Yoshiki
Third Division Department Of Internal Medicine Faculty Of Medicine Kyoto University
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Hattori Ryuichi
Third Division Department Of Internal Medicine Faculty Of Medicine
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Yazaki Yoshio
The Third Dept. Of Medicine University Of Tokyo
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Kawai Chuichi
Third Department Of Internal Medicine Kyoto University Faculty Of Medicine
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OSAKI YASUJI
Dainippon Pharmaceutical Co. Ltd.
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YOHIDA TOMOCHIKA
Ono Pharmaceutical Co. Ltd.
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